Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with Target = 'Histamine H1 receptor' and Ligand = 'BDBM86740'
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  910nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  2.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKd:  2.19E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed