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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Hypoxia-inducible factor prolyl hydroxylase 4 (HIF)' and Ligand = 'BDBM50000403'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Hypoxia-inducible factor prolyl hydroxylase 4 (HIF)


(Homo sapiens (Human))
BDBM50000403
PNG
(5-(2-Carboxy-vinyl)-pyridine-2-carboxylic acid | C...)
Show SMILES OC(=O)\C=C\c1ccc(nc1)C(O)=O
Show InChI InChI=1S/C9H7NO4/c11-8(12)4-2-6-1-3-7(9(13)14)10-5-6/h1-5H,(H,11,12)(H,13,14)/b4-2+
KEGG

UniProtKB/SwissProt

DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 1.06E+4n/an/an/an/an/an/a



ICI Pharmaceuticals

Curated by ChEMBL


Assay Description
Inhibition of prolyl 4-hydroxylase


J Med Chem 35: 800-4 (1992)


Article DOI: 10.1021/jm00083a001
BindingDB Entry DOI: 10.7270/Q25T3M3C
More data for this
Ligand-Target Pair