Affinity DataKi: 19nMAssay Description:Displacement of [3H]diprenorphine from human kappa-opioid receptor expressed in CHO cell membrane for 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Agonist activity at human kappa-opioid receptor expressed in CHO cell membrane assessed as [35S]GTPgammaS binding for 1 hr by liquid scintillation co...More data for this Ligand-Target Pair