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Found 5 Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4A' and Ligand = 'BDBM50158850'
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158850(CHEMBL3785434)
Affinity DataKi:  1.94E+3nMAssay Description:Competitive inhibition of human KDM4A (1 to 359 residues) expressed in competent Escherichia coli BL21-CodonPlus-RIL cells using 2-oxoglutarate as su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158850(CHEMBL3785434)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of KDM4A (unknown origin) measured by antibody-based LANCE Ultra assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158850(CHEMBL3785434)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human KDM4A (1 to 359 residues) expressed in competent Escherichia coli BL21-CodonPlus-RIL cells using H3K9me3 as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158850(CHEMBL3785434)
Affinity DataIC50:  4.66E+4nMAssay Description:Inhibition of human KDM4A (1 to 359 residues) expressed in competent Escherichia coli BL21-CodonPlus-RIL cells using H3K9me3 as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158850(CHEMBL3785434)
Affinity DataIC50:  4.66E+4nMAssay Description:Inhibition of KDM4A (unknown origin) measured by formaldehyde dehydrogenase (FDH)-coupled assayMore data for this Ligand-Target Pair
In DepthDetails PubMed