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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50131241'
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50131241((S)-2-{(S)-2-[(S)-2-(2-Cyano-acetylamino)-3-(3H-im...)
Affinity DataKi:  110nMAssay Description:Binding affinity towards human melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50131241((S)-2-{(S)-2-[(S)-2-(2-Cyano-acetylamino)-3-(3H-im...)
Affinity DataEC50:  18nMAssay Description:In vitro agonist potency was evaluated in HEK293 cells transfected with human melanocortin receptor (hMC4R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed