Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I][Nle4,Dphe7]-alpha-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as stimulation of intracellular cAMP levelMore data for this Ligand-Target Pair