Affinity DataKi: 0.950nMAssay Description:Binding affinity towards human melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]NDP-MSH from Melanocortin 4 receptor at 10 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.510nMAssay Description:Binding affinity towards human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.720nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist potency towards human Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity on mouse melanocortin 4 receptor (mMC4R) stably expressed in HEL cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.720nMAssay Description:effective concentration of peptide at 50% maximal cAMP accumulation on Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity against human melanocortin receptor hMC4RMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0200nMAssay Description:Effective concentration of peptide at 50% maximal cAMP generationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0170nMAssay Description:Evaluated for agonist activity at cloned mammalian Melanocortin 4 receptorMore data for this Ligand-Target Pair