Found 12 Enz. Inhib. hit(s) with Target = 'Melanocyte-stimulating hormone receptor' and Ligand = 'BDBM82411' TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataIC50: 0.510nMAssay Description:Displacement of [125I]NDP-MSH from Melanocortin 1 receptor at 10 uMMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataIC50: 0.510nMAssay Description:Inhibitory concentration against human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataEC50: 0.190nMAssay Description:Effective concentration for intracellular cAMP accumulation in L-cells expressing Melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataEC50: 0.190nMAssay Description:effective concentration of peptide at 50% maximal cAMP accumulation on Melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataEC50: 0.00500nMAssay Description:Decrease in frog skin reflectivity (melanotropic activity).More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataEC50: 0.0700nMAssay Description:Binding affinity towards human melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataEC50: 0.5nMAssay Description:Agonist potency for human Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity on mouse melanocortin 1 receptor (mMC1R) stably expressed in HEK cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataEC50: 0.5nMAssay Description:Agonist activity against human melanocortin receptor hMC1RMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala
Curated by PDSP Ki Database
Uppsala
Curated by PDSP Ki Database
Affinity DataEC50: 0.0230nMAssay Description:Evaluated for agonist activity at cloned mammalian human MSH1 receptorMore data for this Ligand-Target Pair
