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Found 1 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM50181740'
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50181740(2-methoxy-3-[(2-methyl-4-thiazolyl)ethynyl]pyridin...)
Affinity DataIC50:  228nMAssay Description:Activity in agonist-induced phosphoinositide hydrolysis in CHO cells expressing mGluR5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed