Affinity DataKi: 0.319nMAssay Description:Displacement of [3H]methyltrienolone from human mineralocorticoid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.494nMAssay Description:Binding affinity to human mineralocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 27.2nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in HEK293 cells assessed as inhibition of R5050-induced transcriptional activity by...More data for this Ligand-Target Pair