Affinity DataKi: 48nMAssay Description:Binding affinity for human opioid receptor mu 1 using [3H]- DAMGO as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Concentration required to stimulate [35S]GTP-gamma-S, binding to human opioid receptor mu 1 in cell membraneMore data for this Ligand-Target Pair