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Found 3 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50395059'
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50395059(CHEMBL2163917)
Affinity DataKi:  0.274nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50395059(CHEMBL2163917)
Affinity DataIC50:  3.90nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50395059(CHEMBL2163917)
Affinity DataEC50:  0.0342nMAssay Description:Agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30 mins by liqui...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed