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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50033162'
TargetMuscarinic acetylcholine receptor M1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50033162(3-(3-Pentylsulfanyl-pyrazin-2-yl)-1-aza-bicyclo[2....)
Affinity DataIC50:  0.700nMAssay Description:Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]OXO-M as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50033162(3-(3-Pentylsulfanyl-pyrazin-2-yl)-1-aza-bicyclo[2....)
Affinity DataIC50:  1.10nMAssay Description:Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]-Pz as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed