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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Ligand = 'BDBM50208043'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208043(1-methyl-3-(R)-[4,4-Bis-(4-fluoro-phenyl)-2-oxo-im...)
Affinity DataKi:  0.75nMAssay Description:Displacement of [3H]N-methyl-scopalamine from human muscarinic M3 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Via Zambeletti 25

Curated by ChEMBL
LigandPNGBDBM50208043(1-methyl-3-(R)-[4,4-Bis-(4-fluoro-phenyl)-2-oxo-im...)
Affinity DataIC50:  4.5nMAssay Description:Activity at muscarinic M3 receptor in Albino Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed