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Found 1 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Ligand = 'BDBM50345681'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50345681((3-endo)-1,1-Bis-(3-fluorophenyl)-2-(8,8-dimethyl-...)
Affinity DataIC50:  11nMAssay Description:Antagonist activity against human M3 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed