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Found 5 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM48044'
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(3-amino-4,6-dimethyl-N-piperonyl-thieno[2,3-b]pyri...)
Affinity DataKi:  46.8nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(3-amino-4,6-dimethyl-N-piperonyl-thieno[2,3-b]pyri...)
Affinity DataEC50:  403nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(3-amino-4,6-dimethyl-N-piperonyl-thieno[2,3-b]pyri...)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of rat M4 AchRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(3-amino-4,6-dimethyl-N-piperonyl-thieno[2,3-b]pyri...)
Affinity DataEC50:  369nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters

Curated by PubChem BioAssay
LigandPNGBDBM48044(3-amino-4,6-dimethyl-N-piperonyl-thieno[2,3-b]pyri...)
Affinity DataEC50: <1.42E+3nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay