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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50423968'
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423968(CHEMBL2313377)
Affinity DataEC50:  147nMAssay Description:Positive allosteric modulation of rat muscarinic M4 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423968(CHEMBL2313377)
Affinity DataEC50:  77nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO-K1 cells assessed as leftward shift in acetylcholine response treated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed