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Found 4 Enz. Inhib. hit(s) with Target = 'N-alpha-acetyltransferase 50' and Ligand = 'BDBM50541858'
TargetN-alpha-acetyltransferase 50(Homo sapiens)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50541858(CHEMBL4645901)
Affinity DataIC50:  7nMAssay Description:Inhibition of wild type human Naa50 (1852 to 2082 residues) expressed in Escherichia coli BL21(DE3) cells using MLGPEGGEGK peptide as substrate after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-alpha-acetyltransferase 50(Homo sapiens)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50541858(CHEMBL4645901)
Affinity DataKd:  32nMAssay Description:Binding affinity to full length human N-terminal His-tagged/GST-tagged Naa50 expressed in Escherichia coli BL21(DE3) cells in presence of CoA by SPR ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-alpha-acetyltransferase 50(Homo sapiens)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50541858(CHEMBL4645901)
Affinity DataKd:  105nMAssay Description:Binding affinity to full length human N-terminal His-tagged/GST-tagged Naa50 expressed in Escherichia coli BL21(DE3) cells in by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-alpha-acetyltransferase 50(Homo sapiens)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50541858(CHEMBL4645901)
Affinity DataKd:  27nMAssay Description:Binding affinity to full length human N-terminal His-tagged/GST-tagged Naa50 expressed in Escherichia coli BL21(DE3) cells in presence of acetyl CoA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed