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Found 2 Enz. Inhib. hit(s) with Target = 'Na(+)/H(+) exchange regulatory cofactor NHE-RF2' and Ligand = 'BDBM50555257'
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555257(CHEMBL4763464)
Affinity DataKd:  2.82E+3nMAssay Description:Binding affinity to NHERF2 PDZ2 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555257(CHEMBL4763464)
Affinity DataKd:  560nMAssay Description:Binding affinity to NHERF2 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed