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Found 4 Enz. Inhib. hit(s) with Target = 'Orexin receptor type 2' and Ligand = 'BDBM50321510'
TargetOrexin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50321510((3-(7-fluoroquinazolin-2-yl)-3,9-di azabicyclo[4.2...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50321510((3-(7-fluoroquinazolin-2-yl)-3,9-di azabicyclo[4.2...)
Affinity DataKi:  6.70nMAssay Description:Binding affinity to OX2RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50321510((3-(7-fluoroquinazolin-2-yl)-3,9-di azabicyclo[4.2...)
Affinity DataIC50:  136nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50321510((3-(7-fluoroquinazolin-2-yl)-3,9-di azabicyclo[4.2...)
Affinity DataIC50:  150nMAssay Description:Antagonist activity at OX2R by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed