Affinity DataKi: 11nMAssay Description:Binding affinity to human oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [125I]OVTA antagonist from human oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to recombinant oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of [125I]OVTA antagonist from rat oxytocin receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 397nMAssay Description:Binding affinity to oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonism of OT-induced response at OT receptor in rat uterine stripsMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 372nMAssay Description:Compound was evaluated for OT receptor affinity by displacement of [3H]OT from binding sites in uterine tissue taken from nonlabor pregnant womenMore data for this Ligand-Target Pair