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Found 4 Enz. Inhib. hit(s) with Target = 'Phenylethanolamine N-methyltransferase' and Ligand = 'BDBM50072989'
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50072989(1,2,3,4-Tetrahydro-isoquinoline-7-carbonitrile | 1...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro inhibitory activity against bovine adrenal phenylethanolamine N-methyl-transferase (PNMT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50072989(1,2,3,4-Tetrahydro-isoquinoline-7-carbonitrile | 1...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity to human PNMTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50072989(1,2,3,4-Tetrahydro-isoquinoline-7-carbonitrile | 1...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of bovine PNMT by radiochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50072989(1,2,3,4-Tetrahydro-isoquinoline-7-carbonitrile | 1...)
Affinity DataKi:  2.82E+3nMAssay Description:Inhibitory activity against bovine adrenal phenylethanolamine N-methyl-transferase (PNMT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed