BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 2 hits Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4-kinase type 2-alpha' and Ligand = 'BDBM50228494'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Phosphatidylinositol 4-kinase type 2-alpha


(Homo sapiens (Human))
BDBM50228494
PNG
(CHEMBL292541)
Show SMILES Nc1ncnc2n3CCCCc3nc12
Show InChI InChI=1S/C9H11N5/c10-8-7-9(12-5-11-8)14-4-2-1-3-6(14)13-7/h5H,1-4H2,(H2,10,11,12)
PDB

KEGG

UniProtKB/SwissProt

GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
3.58E+4n/an/an/an/an/an/an/an/a



Smith Kline& French Research Limited

Curated by ChEMBL


Assay Description
Binding affinity (Ki) against human phosphatidylinositol 4-kinase


J Med Chem 33: 2073-80 (1990)


Article DOI: 10.1021/jm00170a005
BindingDB Entry DOI: 10.7270/Q25T3NQV
More data for this
Ligand-Target Pair
Phosphatidylinositol 4-kinase type 2-alpha


(Homo sapiens (Human))
BDBM50228494
PNG
(CHEMBL292541)
Show SMILES Nc1ncnc2n3CCCCc3nc12
Show InChI InChI=1S/C9H11N5/c10-8-7-9(12-5-11-8)14-4-2-1-3-6(14)13-7/h5H,1-4H2,(H2,10,11,12)
PDB

KEGG

UniProtKB/SwissProt

GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 5.24E+4n/an/an/an/an/an/a



Smith Kline& French Research Limited

Curated by ChEMBL


Assay Description
Inhibitory activity (IC50) against human phosphatidylinositol 4-kinase at the ATP binding site


J Med Chem 33: 2073-80 (1990)


Article DOI: 10.1021/jm00170a005
BindingDB Entry DOI: 10.7270/Q25T3NQV
More data for this
Ligand-Target Pair