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Compile Data Set for Download or QSAR
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Found
3
Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM27525'
Target
Poly [ADP-ribose] polymerase 1
(Homo sapiens (Human))
Inotek Pharmaceuticals
Ligand
BDBM27525
(N-[3-(morpholin-4-yl)propyl]-8-oxo-9-azatetracyclo...)
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Affinity Data
IC50: 1nM
pH: 8.0 T: 2°C
Assay Description:
The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
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Target
Poly [ADP-ribose] polymerase 1
(Homo sapiens (Human))
Inotek Pharmaceuticals
Ligand
BDBM27525
(N-[3-(morpholin-4-yl)propyl]-8-oxo-9-azatetracyclo...)
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Copy InChI
Affinity Data
IC50: 1nM
Assay Description:
Inhibition of PARP1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Poly [ADP-ribose] polymerase 1
(Homo sapiens (Human))
Inotek Pharmaceuticals
Ligand
BDBM27525
(N-[3-(morpholin-4-yl)propyl]-8-oxo-9-azatetracyclo...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 40nM
Assay Description:
Inhibition of PARP1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI