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Found 4 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50177482'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50177482(1,2,3,11-Tetrahydro-5,11-diaza-benzo[a]trindene-4,...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against human PARP1 expressed in PC12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50177482(1,2,3,11-Tetrahydro-5,11-diaza-benzo[a]trindene-4,...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human recombinant PARP1 in U251MG cells by CometAssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50177482(1,2,3,11-Tetrahydro-5,11-diaza-benzo[a]trindene-4,...)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human PARP1 by in vitro assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50177482(1,2,3,11-Tetrahydro-5,11-diaza-benzo[a]trindene-4,...)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed