Found 12 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily H member 2' and Ligand = 'BDBM50002338' TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 869nMAssay Description:Displacement of [3H]Astemizole from hERG expressed in HEK293 cells at 10 uMMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 33nMAssay Description:Inhibition of hERG K channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 33.2nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 35nMAssay Description:Inhibition of partially open human voltage-gated potassium channel subunit Kv11.1 (ERG K+ channel)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 35.5nMAssay Description:Inhibition of human ERG in MCF7 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 35.7nMAssay Description:K+ channel blocking activity in human embryonic kidney cells expressing HERG Kv11.1More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 95.5nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 191nMAssay Description:Inhibitory concentration against potassium channel HERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 191nMAssay Description:Inhibitory activity against Potassium channel HERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 363nMAssay Description:Inhibition of human Potassium channel HERG expressed in mammalian cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Aventis Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 363nMAssay Description:Inhibition of human ERG expressed in CHO cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
