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Found 4 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50129156'
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129156((Z)-2-(9-fluoro-2,2,4-trimethyl-1,2-dihydrochromen...)
Affinity DataKi:  45nMAssay Description:Inhibitory concentration for antagonistic activity towards human progesterone receptor (hPR) using the cotransfection assay in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129156((Z)-2-(9-fluoro-2,2,4-trimethyl-1,2-dihydrochromen...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]progesterone from Progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129156((Z)-2-(9-fluoro-2,2,4-trimethyl-1,2-dihydrochromen...)
Affinity DataIC50:  65nMAssay Description:Inhibitory concentration for antagonistic activity towards human progesterone receptor (hPR) using the cotransfection assay in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129156((Z)-2-(9-fluoro-2,2,4-trimethyl-1,2-dihydrochromen...)
Affinity DataEC50:  2.70E+3nMAssay Description:Effective concentration for agonist activity towards human progesterone receptor (hPR) using the cotransfection assay in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed