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Found 2 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50010799'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Oregon

Curated by ChEMBL
LigandPNGBDBM50010799(CHEMBL81824 | N-(2-Methyl-4-nitro-phenyl)-N'-o-tol...)
Affinity DataIC50:  37nMAssay Description:In vitro inhibitory activity against [3H]DTG binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Oregon

Curated by ChEMBL
LigandPNGBDBM50010799(CHEMBL81824 | N-(2-Methyl-4-nitro-phenyl)-N'-o-tol...)
Affinity DataIC50:  39nMAssay Description:In vitro inhibitory activity against [3H]- (+)-3-PPP binding to Sigma opioid receptor in guinea pig brain membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed