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Found 2 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50159020'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50159020(4-Benzyl-1-(1,2,3,4-tetrahydro-naphthalen-2-ylmeth...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50159020(4-Benzyl-1-(1,2,3,4-tetrahydro-naphthalen-2-ylmeth...)
Affinity DataKi:  2.52nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed