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Found 3 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM81987'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM81987(CHEMBL116048 | McN-5652-15)
Affinity DataKi:  23.5nMAssay Description:Concentration of the compound inhibiting Dopamine transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Mcneil Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM81987(CHEMBL116048 | McN-5652-15)
Affinity DataKi:  69.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM81987(CHEMBL116048 | McN-5652-15)
Affinity DataKi:  112nMAssay Description:In vitro binding affinity of the compound against Dopamine transporter in LLC-PK1 cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed