Found 7 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50029150'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Mcneil Pharmaceutical
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:In vitro inhibitory constant against [3H]-paroxetine binding to rat frontal cortex membrane serotonin reuptake siteMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Effect of compound on Serotonin transporter uptake from rat cortex using [3H]citalopram as radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Mcneil Pharmaceutical
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Mcneil Pharmaceutical
Curated by PDSP Ki Database
Affinity DataIC50: 10nMAssay Description:Inhibition of uptake of 5-HT in rat brain cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:In vivo inhibition of uptake of 5-HT in human plateletsMore data for this Ligand-Target Pair