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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50088336'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088336(9-(3,4-Dichloro-benzylidene)-7-aza-tricyclo[4.3.1....)
Affinity DataKi:  0.560nMAssay Description:Compound was evaluated for binding affinity using [125I]RTI-55 as a radioligand in HEK-hSERT cells expressing human serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088336(9-(3,4-Dichloro-benzylidene)-7-aza-tricyclo[4.3.1....)
Affinity DataKi:  20nMAssay Description:Inhibition of reuptake of [3H]5-HT at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088336(9-(3,4-Dichloro-benzylidene)-7-aza-tricyclo[4.3.1....)
Affinity DataKi:  20nMAssay Description:Inhibition of reuptake of [3H]5-HT at serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50088336(9-(3,4-Dichloro-benzylidene)-7-aza-tricyclo[4.3.1....)
Affinity DataKi:  30nMAssay Description:Compound was evaluated for inhibition of [3H]5-HT uptake in HEK-hSERT cells expressing Human serotonin transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed