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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50136674'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]RTI-55 from human recombinant SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
The State University Of New York

Curated by ChEMBL
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-dawley rat frontal cortex by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
The State University Of New York

Curated by ChEMBL
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataKi:  8.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of [3H]5HT reuptake at human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed