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Found 5 Enz. Inhib. hit(s) with Target = 'Solute carrier family 15 member 1' and Ligand = 'BDBM50139892'
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University Of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataKi:  180nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University Of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataKi:  1.10E+5nMAssay Description:Binding affinity against membrane transport protein PEPT1 in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University Of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataIC50:  180nMAssay Description:Concentration required to inhibit the maximum [14C]-Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University Of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataIC50:  7.00E+4nMAssay Description:Binding affinity to human PEPT1 assessed as inhibition of [14C]Gly-Sar uptake in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 15 member 1(Homo sapiens (Human))
University Of Tromsø

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataEC50:  1.10E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed