Found 5 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 2' and Ligand = 'BDBM50367247'
TargetSolute carrier family 22 member 2(Homo sapiens (Human))
Anatomisches Institut Der Bayerischen Julius-Maximilians-Universit£T
Curated by ChEMBL
Anatomisches Institut Der Bayerischen Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataKi: 5.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the presence of bicarbonate) (TEA: 20 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the absence of bicarbonate) (TEA: 20 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair