TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKi: 0.0530nMAssay Description:Displacement of [125I]-somatostatin from human SSTR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKi: 0.316nMAssay Description:Binding affinity towards human Somatostatin receptor type 2 (sst2) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKi: 0.501nMAssay Description:Binding affinity for SSTR2 receptors of rat cortex membranes was determined by using [125I][Tyr3]-octreotide radioligandMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Binding affinity for SSTR2 receptors of rat cortex membranes was determined by using Y-labelled SMT487 radioligandMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKd: 0.776nMAssay Description:Binding assay at human somatostatin receptor 2 (hsst2) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKd: 0.610nMAssay Description:Binding affinity to human SST2 receptorMore data for this Ligand-Target Pair