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Found 6 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 2' and Ligand = 'BDBM50272772'
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity towards somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human SSTR2AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50:  0.0200nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(MOUSE)
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50:  0.280nMAssay Description:Tested for inhibition of radioligand binding to cloned somatostatin receptor mSSTR2bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed