Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Sphingosine 1-phosphate receptor 3' and Ligand = 'BDBM50314402'
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50314402((R)-2-amino-2-((S)-6-octyl-1,2,3,4-tetrahydronapht...)
Affinity DataEC50:  97.4nMAssay Description:Agonist activity at human S1P3 receptor assessed as effect on calcium mobilization by Gq dependent whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50314402((R)-2-amino-2-((S)-6-octyl-1,2,3,4-tetrahydronapht...)
Affinity DataEC50:  0.286nMAssay Description:Agonist activity at human S1P3 receptor assessed as effect on calcium mobilization by Gi dependent whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed