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Found 1 Enz. Inhib. hit(s) with Target = 'Stromelysin-1' and Ligand = 'BDBM13134'
TargetStromelysin-1(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM13134((2R)-2-[benzyl(4-methoxybenzene)sulfonamido]-3-cyc...)
Affinity DataKi:  44nMAssay Description:Stromelysin inhibitory activity is based on the hydrolysis of substance P by recombinant human stromelysin to generate a fragment, substance P 7-11, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed