Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50002656'
TargetSubstance-P receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50002656(((2S,3S)-2-Benzyl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2...)
Affinity DataIC50:  234nMAssay Description:Binding affinity was measured against the Tachykinin receptor 1 in CHO-expressed hNK1 using [125I]SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50002656(((2S,3S)-2-Benzyl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2...)
Affinity DataIC50:  487nMAssay Description:Binding affinity towards Tachykinin receptor 1 in human IM-9 cells using [3H]-substance P as ligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed