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Found 2 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50403993'
TargetSubstance-P receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50403993(CHEMBL91418)
Affinity DataKi:  25nMAssay Description:Negative logarithm causing 50% receptor occupancy against tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM50403993(CHEMBL91418)
Affinity DataIC50:  25nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed