Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Trace amine-associated receptor 1' and Ligand = 'BDBM109442'
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
Hoffmann-La Roche

US Patent
LigandPNGBDBM109442(US8604061, 169)
Affinity DataKi:  1.40nMAssay Description:Radioligand binding assay using TAAR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM109442(US8604061, 169)
Affinity DataEC50:  52nMAssay Description:Agonist activity at rat TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
Roche Innovation Center Basel

Curated by ChEMBL
LigandPNGBDBM109442(US8604061, 169)
Affinity DataEC50:  143nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed