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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ITK/TSK' and Ligand = 'BDBM50186460'
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50186460(CHEMBL209148 | N-(5-(5-(1-acetylpiperazine-4-carbo...)
Affinity DataKi:  16nMAssay Description:Inhibition of ITKMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50186460(CHEMBL209148 | N-(5-(5-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human ITK using poly-Glu-Tyr (4:1) as substrate incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50186460(CHEMBL209148 | N-(5-(5-(1-acetylpiperazine-4-carbo...)
Affinity DataIC50:  19nMAssay Description:Inhibition of ItkMore data for this Ligand-Target Pair