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Found 3 Enz. Inhib. hit(s) with Target = 'Vasopressin V1b receptor' and Ligand = 'BDBM301684'
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ferring

US Patent
LigandPNGBDBM301684(US10131692, Compound 16 | US10131692, Compound 27)
Affinity DataEC50:  4.81E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ferring

US Patent
LigandPNGBDBM301684(US10131692, Compound 16 | US10131692, Compound 27)
Affinity DataEC50:  480nMAssay Description:Agonist activity at recombinant human V1B receptor expressed in HEK293 cells measured after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Ferring

US Patent
LigandPNGBDBM301684(US10131692, Compound 16 | US10131692, Compound 27)
Affinity DataEC50:  1.33E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent