Found 2 Enz. Inhib. hit(s) with Target = 'Voltage-dependent L-type calcium channel subunit alpha-1S' and Ligand = 'BDBM50479922'
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universita Degli Studi Di Bologna
Curated by ChEMBL
Universita Degli Studi Di Bologna
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel in Sprague-Dawley rat cardiac myocytes by liquid scintillation countingMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Universita Degli Studi Di Bologna
Curated by ChEMBL
Universita Degli Studi Di Bologna
Curated by ChEMBL
Affinity DataIC50: 3.34E+4nMAssay Description:Inhibition of L-type calcium channel in Wistar rat tail artery smooth muscle cells assessed as blockade of barium-sensitive inward rectifying current...More data for this Ligand-Target Pair