Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for monomerid = 10452
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  126nMAssay Description:Binding affinity to human alpha1A adrenergic receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]-prazosin from human alpha1A adrenergic receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  148nMAssay Description:Binding affinity to human alpha1B adrenergic receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]-prazosin from human alpha1B adrenergic receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]-prazosin from human alpha1D adrenergic receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  309nMAssay Description:Binding affinity to human alpha1D adrenergic receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  832nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM10452(Bivalent 4-Aminoquinoline 9f | N,N-di-4-Quinolyl-1...)
Affinity DataKi:  832nMAssay Description:Binding affinity to human 5HT1A receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed