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Found 6 of ic50 for monomerid = 10842
LigandPNGBDBM10842(3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol | ...)
Affinity DataIC50:  90nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Cnrs

LigandPNGBDBM10842(3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol | ...)
Affinity DataIC50:  150nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM10842(3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol | ...)
Affinity DataIC50:  180nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Rattus norvegicus (rat))
Cnrs

LigandPNGBDBM10842(3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol | ...)
Affinity DataIC50:  400nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase 1(Bos taurus (bovine))
Cnrs

LigandPNGBDBM10842(3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol | ...)
Affinity DataIC50:  600nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Cnrs

LigandPNGBDBM10842(3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol | ...)
Affinity DataIC50:  2.50E+3nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed