Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ki for monomerid = 113119
TargetKallikrein-7(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi:  80nM ΔG°:  -10.1kcal/molepH: 7.2 T: 2°CAssay Description:Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi: <100nM ΔG°: <-9.93kcal/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProthrombin(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi:  600nM ΔG°:  -8.82kcal/molepH: 8.3 T: 2°CAssay Description:Materials: Thrombin (Chromogenics, cat. no. 820712), Substrate S-2288 (Chromogenics, cat. no. 82 08 52). Thrombin activity was determined at 37° ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCathepsin G(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi:  700nM ΔG°:  -8.73kcal/molepH: 7.2 T: 2°CAssay Description:Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi:  1.00E+3nM ΔG°:  -8.51kcal/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetKallikrein-14(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi:  1.40E+3nM ΔG°:  -8.30kcal/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK14, Substrate S-2302 (Chromogenics, cat. no. 820340). KLK14 activity was determined at 37° C. in 0.1 mM Tris, pH ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi: >1.00E+4nM ΔG°: >-7.09kcal/molepH: 7.2 T: 2°CAssay Description:Materials: Trypsin, 100 ug (Roche, sequence grade, Mw 23500), Substrate S-2288 (Chromogenics, cat. no. 820852). Trypsin activity was determined at 3...More data for this Ligand-Target Pair
In DepthDetails US Patent