Affinity DataKi: 0.5nM ΔG°: -11.8kcal/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]PK11195 from translocator protein in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat kidney mitochondrial membranes by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to peripheral benzodiazepine receptors using [3H]-PK11195 radioligand in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H]-flunitrazepam from TSPO receptor in Wistar rat brain without cerebellum incubated for 90 mins by liquid scintillation counter an...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
Georgetown University
Curated by PDSP Ki Database
Georgetown University
Curated by PDSP Ki Database