Found 22 of ec50 for monomerid = 22496 
Affinity DataEC50: 79nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair
Affinity DataEC50: 99nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at FFAR1 (unknown origin) assessed as increase in ERK1/2 MAP kinase phosphorylationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at human GPR40 H86F mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human GPR40 H137A mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Agonist activity at human GPR40 H86A mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
Affinity DataEC50: 6.80E+3nMAssay Description:Agonist activity at human GPR40 H137F mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
Affinity DataEC50: 1.78E+4nMAssay Description:Agonist activity at human GPR40 N244A mutant expressed in HEK-EM 293 cells assessed as increase in intracellular calciumMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Agonist activity at human C-terminal eYFP-tagged FFA1 receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment incubated for 5 mins...More data for this Ligand-Target Pair
Affinity DataEC50: 28.2nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 1.41E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataEC50: 47.9nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells assessed as calcium mobilization by fluorescence spectrophotometryMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
Affinity DataEC50: 47.9nMAssay Description:Agonist activity at human FFA1 expressed in CHO cells by Gal4 luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells after 24 hrs by NFAT-luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 3.50E+3nMAssay Description:Agonist activity at human GPR120 expressed in baculovirus infected sf9 cells assessed as increase in calcium flux measured every 1 sec for 60 secs by...More data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as increase in calcium flux measured every 2 secs for 90 secs by Calcium-3 dye bas...More data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Agonist potency at human GPR40 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human FFA1 expressed in HEK293 cells assessed as stimulation of intracellular calcium mobilization measured at 2 secs time interv...More data for this Ligand-Target Pair
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human FFA4 expressed in HEK293 cells assessed as stimulation of intracellular calcium mobilization measured at every 1 secs for 6...More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
